György Miklós Keserű - Selected Publications#


1. Pandy-Szekeres, Gaspar; Caroli, Jimmy; Mamyrbekov, Alibek; Kermani, Ali A.; Keseru, Gyorgy M.; Kooistra, Albert J.; Gloriam, David E. GPCRdb in 2023: state-specific structure models using AlphaFold2 and new ligand resources
NUCLEIC ACIDS RESEARCH 51: D1 pp. D395-D402., 8 p. (2022)

2. Bajusz, Dávid; Wade, Warren S.; Satała, Grzegorz; Bojarski, Andrzej J.; Ilaš, Janez; Ebner, Jessica; Grebien, Florian; Papp, Henrietta; Jakab, Ferenc; Douangamath, Alice et al. Keserű, György M Exploring protein hotspots by optimized fragment pharmacophores
NATURE COMMUNICATIONS 12: 1 Paper: 3201 (2021)

3. Kooistra, Albert J; Mordalski, Stefan; Pándy-Szekeres, Gáspár; Esguerra, Mauricio; Mamyrbekov, Alibek; Munk, Christian; Keserű, György M; Gloriam, David E GPCRdb in 2021: integrating GPCR sequence, structure and function
NUCLEIC ACIDS RESEARCH 49: D1 pp. D335-D343. (2021)

4. Prokop, Susanne; Ábrányi-Balogh, Péter; Barti, Benjámin; Vámosi, Márton; Zöldi, Miklós; Barna, László; Urbán, Gabriella M.; Tóth, András Dávid; Dudok, Barna; Egyed, Attila; Keseru, Gyorgy M. et al. PharmacoSTORM nanoscale pharmacology reveals cariprazine binding on Islands of Calleja granule cells
NATURE COMMUNICATIONS 12: 1 Paper: 6505 , 19 p. (2021)

5. Szabó, György; Erdélyi, Péter; Kolok, Sándor; Vastag, Mónika; Halász, Attila S.; Kis-Varga, Istvánné; Lévay, György I.; Béni, Zoltán; Kóti, János; Greiner, István; Keseru, Gyorgy M. et al. Fragment-Based Optimization of Dihydropyrazino-Benzimidazolones as Metabotropic Glutamate Receptor-2 Positive Allosteric Modulators against Migraine
JOURNAL OF MEDICINAL CHEMISTRY 64: 12 pp. 8607-8620. , 14 p. (2021)

6. Douangamath, Alice; Fearon, Daren; Gehrtz, Paul; Krojer, Tobias; Lukacik, Petra; Owen, C. David; Resnick, Efrat; Strain-Damerell, Claire; Aimon, Anthony; Abranyi-Balogh, Peter; Keseru, Gyorgy M. et al. Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease
NATURE COMMUNICATIONS 11: 1 Paper: 5047 , 11 p. (2020)

7. Egyed, Attila; Domány-Kovács, Katalin; Koványi, Bence; Horti, Ferenc; Kurkó, Dalma; Kiss, Dóra Judit; Pándy-Szekeres, Gáspár; Greiner, István; Keserű, György M. Controlling receptor function from the extracellular vestibule of G-protein coupled receptors
CHEMICAL COMMUNICATIONS 56: 91 pp. 14167-14170., 4 p. (2020)

8. Menyhard, Dora K.; Palfy, Gyula; Orgovan, Zoltan; Vida, Istvan; Keseru, Gyorgy M.; Perczel, Andras Structural impact of GTP binding on downstream KRAS signaling
CHEMICAL SCIENCE 11: 34 pp. 9272-9289., 18 p. (2020)

9. Egbert, Megan; Whitty, Adrian; Keserű, György M.; Vajda, Sandor Why Some Targets Benefit from beyond Rule of Five Drugs
JOURNAL OF MEDICINAL CHEMISTRY 62: 22 pp. 10005-10025. Paper: acs.jmedchem.8b01732, 21 p. (2019)

10. Boström, J.; Brown, D.G.; Young, R.J. ; Keserü, G.M. Expanding the medicinal chemistry synthetic toolbox
NATURE REVIEWS DRUG DISCOVERY 17: 10 pp. 709-727., 19 p. (2018)

Web of Science:

Publications: 314
Times Cited: 7349
H-Index: 42

Google ScholarAllSince 2018
Citations 123575347
h-index5231
i10-index18395

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