Cesare Gennari - Publications#


H index (Scopus): 46 (5/12/2020)
Total citations (Scopus): 7.779 (5/12/2020)

Selected Publications

1) Fast Cyclization of a Proline-Derived Self-Immolative Spacer Improves the Efficacy of Carbamate Prodrugs
Dal Corso, A.; Borlandelli, V.; Corno, C.; Perego, P.; Belvisi, L.; Pignataro, L.; Gennari, C.
Angew. Chem. Int. Ed. 2020, 59, 4176-4181; DOI: 10.1002/anie.201916394

2) Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake
Pina, A.; Kadri, M.; Arosio, D.; Dal Corso, A.; Coll, J.-L.; Gennari, C.; Boturyn, D.
Chemistry - A European Journal 2020, 26, 7492-7496; DOI: 10.1002/chem.202001115

3) Innovative linker strategies for tumor-targeted drug conjugates
Dal Corso, A.; Pignataro, L.; Belvisi, L.; Gennari, C.
Chemistry - A European Journal 2019, 25, 14740-14757; DOI: 10.1002/chem.201903127

4) Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate
Raposo Moreira Dias, A.; Pina, A.; Dean, A.; Lerchen, H.-G.; Caruso, M.; Gasparri, F.; Fraietta, I.; Troiani, S.; Arosio, D.; Belvisi, L.; Pignataro, L.; Dal Corso, A.; Gennari, C.
Chemistry - A European Journal 2019, 25, 1696-1700; DOI: 10.1002/chem.201805447

5) Efficient Synthesis of Amines by Iron-Catalyzed C=N Transfer Hydrogenation and C=O Reductive Amination
Vailati Facchini, S.; Cettolin, M.; Bai, X.; Casamassima, G.; Pignataro, L.; Gennari, C.; Piarulli, U.
Adv. Synth. Catal. 2018, 360, 1054-1059; DOI 10.1002/adsc.201701316

6) Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin aVb3
Raposo Moreira Dias, A.; Pina, A.; Dal Corso, A.; Arosio, D.; Belvisi, L.; Pignataro, L.; Caruso, M.; Gennari, C.
Chemistry - A European Journal 2017, 23, 14410-14415; DOI: 10.1002/chem.201703093

7) Tumor Targeting with an isoDGR-Drug Conjugate
Zanella, S.; Angerani, S.; Pina, A.; López Rivas, P.; Giannini, C.; Panzeri, S.; Arosio, D.; Caruso, M.; Gasparri, F.; Fraietta, I.; Albanese, C.; Marsiglio, A.; Pignataro, L.; Belvisi, L.; Piarulli, U.; Gennari, C.
Chemistry - A European Journal 2017, 23, 7910-7914; DOI: 10.1002/chem.201701844

8) Asymmetric Transfer Hydrogenation of Ketones with modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process
Renom-Carrasco, M.; Gajewski, P.; Pignataro, L.; de Vries, J. G.; Piarulli, U.; Gennari, C.; Lefort, L.
Adv. Synth. Catal. 2016, 358, 515-519; DOI: 10.1002/adsc.201500933

9) Asymmetric Hydrogenation of 3-Substituted Pyridinium Salts
Renom-Carrasco, M.; Gajewski, P.; Pignataro, L.; de Vries, J. G.; Piarulli, U.; Gennari, C.; Lefort, L.
Chemistry - A European Journal 2016, 22, 9528-9532; DOI: 10.1002/chem.201601501

10) Mixed Ligand Approach for the Asymmetric Hydrogenation of 2-Substituted Pyridinium Salts
Renom-Carrasco, M.; Gajewski, P.; Pignataro, L.; de Vries, J. G.; Piarulli, U.; Gennari, C.; Lefort, L.
Adv. Synth. Catal. 2016, 358, 2589-2593; DOI: 10.1002/adsc.201600348

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